| 2,4-dinitrophenol |
24 hr |
100μM |
High |
| 2-nitrofluorene |
24 hr |
100μM |
High |
| acarbose |
24 hr |
2000μM |
Middle |
| acetamide |
8 hr |
10000μM |
High |
| acetamidofluorene |
24 hr |
50μM |
High |
| acetaminophen |
24 hr |
200μM |
Low |
| acetazolamide |
8 hr |
120μM |
Middle |
| adapin |
24 hr |
75μM |
High |
| aflatoxin B1 |
24 hr |
6μg/mL |
High |
| ajmaline |
24 hr |
300μM |
High |
| allopurinol |
24 hr |
140μM |
High |
| allyl alcohol |
8 hr |
14μM |
Middle |
| alpidem |
24 hr |
10μM |
High |
| amiodarone |
2 hr |
7μM |
High |
| amitriptyline |
24 hr |
15μM |
High |
| amphotericin B |
24 hr |
2μM |
High |
| aspirin |
2 hr |
600μM |
Middle |
| azathioprine |
24 hr |
14.6μM |
Middle |
| bendazac |
8 hr |
40μM |
Middle |
| benzbromarone |
24 hr |
100μM |
High |
| benziodarone |
8 hr |
8μM |
Middle |
| bromobenzene |
2 hr |
40μM |
Middle |
| bromoethylamine |
24 hr |
500μM |
High |
| bucetin |
8 hr |
60μM |
Middle |
| buspirone |
24 hr |
30μM |
High |
| buthionine sulfoximine |
24 hr |
10000μM |
High |
| butylated hydroxyanisole |
24 hr |
200μM |
High |
| caffeine |
24 hr |
7500μM |
High |
| captopril |
24 hr |
8000μM |
High |
| carbamazepine |
8 hr |
12μM |
Low |
| carbon tetrachloride |
8 hr |
7500μM |
High |
| chloramphenicol |
8 hr |
90μM |
Middle |
| chlormadinone |
24 hr |
8μM |
Middle |
| chlormezanone |
24 hr |
250μM |
High |
| chlorpheniramine |
24 hr |
90μM |
High |
| chlorpromazine |
24 hr |
20μM |
High |
| chlorpropamide |
24 hr |
750μM |
High |
| cimetidine |
8 hr |
60μM |
Middle |
| ciprofloxacin |
24 hr |
25μM |
High |
| clofibrate |
2 hr |
60μM |
Middle |
| clomipramine |
8 hr |
10μM |
High |
| clozapine |
24 hr |
50μM |
High |
| colchicine |
8 hr |
800μM |
Middle |
| coumarin |
2 hr |
300μM |
High |
| cycloheximide |
24 hr |
100μM |
High |
| cyclophosphamide |
2 hr |
400μM |
Middle |
| cyclosporine A |
24 hr |
6μM |
High |
| danazol |
8 hr |
35μM |
High |
| dantrolene |
24 hr |
2μM |
Middle |
| dexamethasone |
8 hr |
12μM |
Low |
| diazepam |
2 hr |
250μM |
High |
| diclofenac |
2 hr |
80μM |
Middle |
| diethyl maleate |
8 hr |
1500μM |
High |
| diltiazem |
24 hr |
150μM |
High |
| disopyramide |
24 hr |
3500μM |
High |
| disulfiram |
24 hr |
12μM |
Middle |
| doxorubicin |
24 hr |
10μM |
High |
| enalapril |
24 hr |
2000μM |
High |
| erythromycin ethylsuccinate |
24 hr |
5μM |
High |
| ethambutol |
24 hr |
4000μM |
High |
| ethanol |
24 hr |
10000μM |
High |
| ethinylestradiol |
8 hr |
3μM |
Middle |
| ethionamide |
8 hr |
120μM |
Middle |
| ethionine |
24 hr |
400μM |
Low |
| etoposide |
24 hr |
330μM |
High |
| famotidine |
8 hr |
140μM |
Middle |
| fenofibrate |
24 hr |
6μM |
Middle |
| fluoxetine hydrochloride |
24 hr |
20μM |
High |
| fluphenazine |
24 hr |
4μM |
Middle |
| flutamide |
2 hr |
50μM |
High |
| furosemide |
8 hr |
500μM |
Middle |
| galactosamine |
24 hr |
10000μM |
High |
| gemfibrozil |
2 hr |
100μM |
High |
| glibenclamide |
2 hr |
4μM |
Middle |
| griseofulvin |
8 hr |
4μM |
Middle |
| haloperidol |
2 hr |
4μM |
Middle |
| hepatocyte growth factor, human |
8 hr |
10ng/mL |
Middle |
| hexachlorobenzene |
2 hr |
30μM |
High |
| hydroxyzine |
24 hr |
40μM |
High |
| ibuprofen |
24 hr |
150μM |
High |
| imipramine |
24 hr |
15μM |
High |
| indomethacin |
8 hr |
200μM |
High |
| interferon alpha, human |
2 hr |
2ng/mL |
Low |
| interleukin 1 beta, human |
2 hr |
2ng/mL |
Low |
| interleukin 6, human |
2 hr |
10ng/mL |
Middle |
| iproniazid |
24 hr |
1200μM |
High |
| isoniazid |
2 hr |
2000μM |
Middle |
| ketoconazole |
8 hr |
0.6μM |
Low |
| labetalol |
2 hr |
5.6μM |
Low |
| lomustine |
8 hr |
24μM |
Middle |
| lornoxicam |
24 hr |
3μM |
Middle |
| mefenamic acid |
8 hr |
30μM |
Middle |
| meloxicam |
8 hr |
50μM |
High |
| metformin |
8 hr |
200μM |
Middle |
| methapyrilene |
2 hr |
24μM |
Low |
| methimazole |
8 hr |
10000μM |
High |
| methyldopa |
8 hr |
10μM |
Middle |
| methylene dianiline |
24 hr |
24μM |
Low |
| methyltestosterone |
2 hr |
4μM |
Middle |
| mexiletine |
24 hr |
300μM |
High |
| monocrotaline |
8 hr |
18μM |
Middle |
| moxisylyte |
24 hr |
400μM |
High |
| naphthyl isothiocyanate |
24 hr |
200μM |
High |
| naproxen |
24 hr |
600μM |
High |
| nefazodone |
24 hr |
30μM |
High |
| nicotinic acid |
8 hr |
2000μM |
Middle |
| nifedipine |
8 hr |
150μM |
High |
| nimesulide |
24 hr |
330μM |
High |
| nitrofurantoin |
2 hr |
5μM |
Low |
| nitrofurazone |
24 hr |
50μM |
High |
| nitrosodiethylamine |
24 hr |
2000μM |
Middle |
| omeprazole |
2 hr |
120μM |
Middle |
| papaverine |
24 hr |
60μM |
High |
| pemoline |
24 hr |
75μM |
High |
| penicillamine |
24 hr |
10000μM |
High |
| perhexiline |
24 hr |
15μM |
High |
| phalloidin |
8 hr |
80μg/mL |
Middle |
| phenacetin |
24 hr |
600μM |
High |
| phenobarbital |
8 hr |
400μM |
Low |
| phenylanthranilic acid |
24 hr |
40μM |
Middle |
| phenylbutazone |
2 hr |
16μM |
Low |
| phenytoin |
24 hr |
2.4μM |
Low |
| phorone |
8 hr |
5000μM |
High |
| promethazine |
24 hr |
35μM |
High |
| propranolol |
24 hr |
100μg/kg |
High |
| propylthiouracil |
2 hr |
4000μM |
High |
| quinidine |
24 hr |
50μM |
High |
| ranitidine |
24 hr |
4000μM |
High |
| rifampicin |
8 hr |
70μM |
High |
| rosiglitazone maleate |
8 hr |
12μg/kg |
Low |
| rotenone |
8 hr |
2μM |
High |
| simvastatin |
8 hr |
30μM |
High |
| sulfasalazine |
8 hr |
150μM |
High |
| sulindac |
8 hr |
600μM |
Middle |
| sulpiride |
24 hr |
1000μM |
Middle |
| tacrine |
24 hr |
80μM |
High |
| tamoxifen |
8 hr |
25μM |
High |
| tannic acid |
8 hr |
1μM |
Middle |
| terbinafine |
24 hr |
15μM |
High |
| tetracycline |
8 hr |
5μM |
Middle |
| theophylline |
24 hr |
10000μM |
High |
| thioacetamide |
2 hr |
10000μM |
High |
| thioridazine |
24 hr |
15μM |
High |
| ticlopidine |
24 hr |
20μM |
High |
| tiopronin |
8 hr |
400μM |
Middle |
| tolbutamide |
8 hr |
400μM |
Middle |
| transforming growth factor beta 1 |
8 hr |
50ng/mL |
High |
| triazolam |
24 hr |
0.4μM |
Low |
| trimethadione |
8 hr |
2000μM |
Middle |
| tunicamycin |
8 hr |
10μg/mL |
High |
| valproic acid |
2 hr |
200μM |
Low |
| venlafaxine |
24 hr |
1200μM |
High |
| vitamin A |
24 hr |
7.5μM |
High |
| LPS |
24 hr |
60μg/mL |
Middle |
| N-methyl-N-nitrosourea |
8 hr |
10000μM |
High |
| N-nitrosomorpholine |
24 hr |
10000μM |
High |
| TNFa |
24 hr |
50ng/mL |
High |
| WY-14643 |
8 hr |
6μM |
Low |